In this study, it is clear from the in vitro inhibition kinetic studies in rat liver microsomes that MA can act as competitive inhibitor
to rat CYP2C11 with a of 98.
Perchlorate is a competitive inhibitor
of the sodium iodide symporter (NIS), the thyroid cell-surface protein responsible for transporting iodide from the plasma into the thyroid.
Dihydrotanshinone was not only a potent competitive inhibitor
of human CYP1A2 and CYP2C9, but also a potent noncompetitive inhibitor of human CYP3A4.
Tricyclic antidepressants block the reuptake of serotonin and norepinephrine, are competitive inhibitors
Oseltamivir and zanamivir are competitive inhibitors
for the neuraminidase enzyme for the influenza virus.
Current approaches to neutralising chemoresistance have centred on developing competitive inhibitors