The screening of all the synthesized compounds against butyrylcholinesterase enzyme revealed that only three compounds showed good activity, N-benzyl-N-(3-hydroxyphenyl)-2,3-dihydrobenzo[1,4]dioxine-6-sulfonamide (6c), N-benzyl-2,3-dihydrobenzo[1,4]dioxine-6-sulfona-mide (3d), N-benzyl-N-(3,5-dimethylphenyl)-2,3-dihydrobenzo [1,4] dioxine-6-sulfonamide (6a) having IC50 values of 71.27+-0.01, 198.21+-0.11 and 259.61+-0.01 umoles/L respectively, comparative to
eserine (Table 2).
Eserine salt was used as the positive standard, and the dilutions of both the samples and the standard were based on a concentration of 20mg x [mL.sup.-1] [19, 20].
Eserine (0.5 mM well-1) was used as positive control.
Although bands of both strains exhibited equal affinity, bands E-11 and E-12 in both strains were classified as
eserine sulfate sensitive carboxylesterasae (Owusa et al., 1996).
D: Complete the words
ESERINE, EMINENT, POLITIC and INDENES in that order.
The results suggest that the studied enzymes are ChEs and not nonspecific esterases, due to their apparent affinity for choline esters, with a distinct preference for the substrate acetyl-thiocholine, and their high sensitivity to inhibition by
eserine sulfate.
Paminetinas ir iki siol Nidoje islikes restoranas "
Eserine" (1979 m., arch.
Administration of carbachol, acetylcholine or pilocarpine into AMR and DMV elicited dose-related decreases in heart rate, similarly
eserine injected into these nuclei augmented and prolonged the action of acetylcholine.
Burada dikkat edilmesi gereken nokta 'Yablo 1992' (bir esere referans verir) ve 'Yablo (1992)' (bir yazara ve parantez icinde onun bir
eserine referans verir) arasindaki farktir.
Bu makalede, on dokuzuncu yuzyilin sonunda kavram olarak ortaya atilmasindan itibaren sekillendirilen mazosizmin bircok tanimi ele alinarak Bram Stoker'in Dracula adli
eserine uygulanmistir.
Bu dusunceyle hareket eden sairin, yazdigi
eserine karsilik devlet ricalinden ya da varlikli kisilerden caize alabilmesi icin o kisilere eserini takdim etmesi gerekir.